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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T5203 | Sodium Tartrate | Others | |
Sodium Tartrate is a food additive, used as an emulsifier and binding agent in food products. | |||
TN7074 | (2E)-3-(1,3-Benzodioxol-5-yl)-2-propenoic acid | Antibiotic | |
(2E)-3-(1,3-Benzodioxol-5-yl)-2-propenoic acid displays EC50 values of 73.5 μM against T. cruzi. trypomastigotes. | |||
T9494 | Imidazole-5-propionic acid | Imidazolylpropionic acid,SALOR-INT L480258-1EA,Deamino-histidine | Dehydrogenase |
Imidazole-5-propionic acid (Imidazolylpropionic acid) is a product of histidine metabolism and may involve oxidation or transamination. Imidazole-5-propionic acid is potent inhibitors of G. candidum histidinol dehydrogen... | |||
TN1258 | 3-Acetyl-beta-boswellic acid | 3-O-Acetyl-beta-boswellic acid | DNA/RNA Synthesis |
3-Acetyl-beta-boswellic acid has antitumor activity, it inhibits synthesis of DNA, RNA and protein in human leukemia HL-60 cells in a dose dependent manner with IC50 values ranging from 0.6 to 7.1 microM. | |||
T77557 | Coumarin343 | ||
Coumarin343 inhibits monocarboxylic acid transporter protein 4 with IC50 values in the range of 0.01-100 µM.Coumarin343 exhibits anticancer and antibacterial activity.Coumarin343 is a coumarin dye. | |||
T10017 | 1-Linoleoyl Glycerol | Glycerol 1-monolinolate,Monolinolein,Glyceryl monolinoleate,1-Linoleoyl-rac-glycerol | Phospholipase |
1-Linoleoyl Glycerol (Monolinolein) is fatty acid glycerol that has been isolated from Saururus Chinensis roots. The (R)-1-Linoleoyl Glycerol and (S)-1-Linoleoyl Glycerol exhibit Lipoprotein-associated phospholipase A2 (... | |||
T11888 | LtaS-IN-1 | Others , Antibacterial | |
LtaS-IN-1 is an effective inhibitor of Lipoteichoic acid synthesis in multidrug-resistant (MDR) E. faecium and by altering the cell wall morphology. LtaS-IN-1 is against Enterococcus spp 28 strains with varying MIC value... | |||
T12408 | Perhexiline maleate | Others , Mitochondrial Metabolism | |
Perhexiline maleate is an orally active inhibitor of CPT1 and CPT2 that reduces fatty acid metabolism. The IC50 values of perhexiline maleate against rat heart and liver CPT 1 were 77 and 148 μM, respectively. | |||
TCS1372 | Atraric acid | Phosphatase , Androgen Receptor | |
Atraric acid derivatives as a new chemical lead structure for novel therapeutic compounds as AR antagonists, that can be used for prophylaxis or treatment of prostatic diseases. It inhibits PTP1B activity in a dose-depen... | |||
T11363 | Ganoderic acid F | Others | |
Ganoderic acid F exhibits antitumor and antimetastatic activities through inhibition of angiogenesis and alteration of proteins involving cell proliferation and/or cell death, carcinogenesis, oxidative stress, calcium si... | |||
TN2330 | Phenethyl ferulate | Caffeic Acid 3-Methyl Phenethyl Ester | Lipoxygenase , COX |
Phenethyl ferulate (Caffeic Acid 3-Methyl Phenethyl Ester) has chemopreventive properties against chemically induced colon carcinogenesis. It enhances apoptosis in azoxymethane induced colon tumors. It shows inhibitory a... | |||
T39647 | BMS-986278 | LPA Receptor | |
BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb values of 6.9 nM and 4.0 nM for human and mouse LPA1, respectively.BMS-986278 may be investigated for use in idiopathic... | |||
T38905 | FATP1-IN-1 | FATP1-IN-1 | Others |
FATP1-IN-1 is a potent inhibitor of fatty acid transport protein 1 (FATP1). It effectively inhibits the activity of recombinant human or mouse acyl-CoA synthetase, which is essential for the function of FATP1. The inhibi... | |||
TP1930L1 | Spexin acetate(1370290-58-6 free base) | Neuropeptide Y Receptor | |
Spexin acetate is a potent galanin receptor 2/3 (GAL2/GAL3) agonist (EC50 values are 45.7 and 112.2 nM, respectively). Exhibits no significant activity at galanin receptor 1. Endogenous satiety-inducing peptide; inhibits... | |||
T7057 | Methylstat | Histone Demethylase , Others | |
Methylstat is a methyl ester prodrug of a Jumonji C domain-containing histone demethylase (JMJD) inhibitor that has favorable cell permeability. The free acid of methylstat inhibits JMJD2A, JMJD2C, JMJD2E, PHF8, and JMJD... | |||
T21831 | UCM05 | G28UCM | Fatty Acid Synthase |
UCM05 (G28UCM) is a potent inhibitor of fatty acid synthase (FASN) with efficacy against HER2+ breast cancer xenografts, including in cell lines resistant to anti-HER2 drugs [1]. Additionally, it functions as an inhibito... | |||
T38037 | Caffeic Acid-13C3 | Caffeic Acid-13C3 | |
Caffeic acid-13C3 is an isotopically enriched form of caffeic acid that is intended for use as an internal standard for the quantification of caffeic acid by GC- or LC-MS. Caffeic acid is an inhibitor of 5-LO , with IC50... | |||
TN6604 | 4-Chlorocinnamic acid | ||
4-Chlorocinnamic acid is a photosensitive compound. 2-Chlorocinnamic acid and 4-chlorocinnamic acid show potent urease inhibitory activities with the respective IC50 values of 0.66 and 1.10 uM. | |||
T4131 | Arjunic acid | COX , Antifection | |
Arjunic acid is a strong antioxidant and a free radical scavenger. Arjunic acid shows activity against Gram-positive and Gram-negative bacteria with MIC values ranging between 1.9 and 15.6 microg/mL. | |||
TN6659 | 2-Chlorocinnamic acid | ||
2-Chlorocinnamic acid is a photosensitive compound, it can inhibit tyrosinase activity. 2-Chlorocinnamic acid and 4-chlorocinnamic acid show potent urease inhibitory activities with the respective IC50 values of 0.66 and... |